NEWS & TOPICS
Chem. Pharm. Bull. Vol. 72 No. 7
2024/09/02
Cover
Structure-Activity Relationship Study of CYM51010, an Agonist for the μ-δ Opioid Receptor Heterodimer
pp. 711-730
Structure-Activity Relationship Study of CYM51010, an Agonist for the μ-δ Opioid Receptor Heterodimer
pp. 711-730

Current Topics - Frontiers in Alzheimer's and Dementia Research
Foreword
Ken-ichi KusakabeCurrent Topics: Review
Anti-amyloid-β Antibodies and Anti-tau Therapies for Alzheimer's Disease: Recent Advances and Perspectives
Naoyuki Suzuki, Takuya Hatta, Mana Ito, and Ken-ichi Kusakabe
Clinical Pipelines for Alzheimer's Disease Psychosis and Agitation
Takuya Oguma and Kohei Jino
Neuroimmune Dysfunction in Alzheimer's Disease and Other Forms of Dementia
Takuya Yamane, Takeshi Yoshioka, and Yusuke Shimo
Epigenetic Inhibitors as Alzheimer's Disease Therapeutic Agents
Yasunobu Yamashita, Yukihiro Itoh, Yuri Takada, and Takayoshi Suzuki
Current Topics: Regular Article
Identification of Proteolysis Targeting Chimeras (PROTACs) for Lysine Demethylase 5 and Their Neurite Outgrowth-Promoting Activity
Tetsuya Iida, Yukihiro Itoh, Yukari Takahashi, Yuka Miyake, Farzad Zamani, Yasunobu Yamashita, Yuri Takada, Toshiki Akiyama, Jun Ibaraki, Kyoka Okuda, Yuto Tokuda, Tomoka Nishimura, Koto Hidaka, Hiiro Mori, Makoto Oba, and Takayoshi Suzuki
Regular Article
Spectral and HPLC Analyses of Synthesized Butin and Butein
Takashi Kamei, Jun Miyazaki, Ryoga Hori, Hiroaki Saito, Tatsuo Takahashi, Ken-ichi Shinohara, Masakazu Miura, and Hirokazu Suzuki
The Application of Microsampling Disks in Circular Dichroism Spectroscopy for Peptide and Nucleic Acid Drugs
Genichiro Tsuji, Takashi Misawa, and Yosuke Demizu
Note
Estimation for Raw Material Plants of a Henna Product Using LC-High Resolution MS and Multivariate Analysis
Naohiro Oshima, Maiko Tahara, Tsuyoshi Kawakami, Akiko Yagami, Takumi Akiyama, Nahoko Uchiyama, and Yoshiaki Ikarashi
Regular Article
Galangin Promotes Tendon Repair Mediated by Tendon-Derived Stem Cells through Activating the TGF-β1/Smad3 Signaling Pathway
Xiongwei Deng, Qiang Li, Haitao Yuan, Hejun Hu, and Shaoyong Fan
Note
Continuous Monitoring of Pseudopolymorphic Transition in Ezetimibe Using T1 Relaxation with Time-Domain NMR
Takashi Ono, Kotaro Okada, Misaki Kaga, Hidekatsu Eto, Shungo Kumada, Nobuyuki Wakui, and Yoshinori Onuki
Regular Article
Preparation and Evaluation of Clarithromycin Taste-Masking Dry Suspension Using Hot Melt Extrusion Based on Solid Dispersion Technology
Tianao Zhang, Min Yu, Yong Fan, Lingyang Wang, Lu Yuan, and Yong Sun
Note
Total Synthesis of Dinorsesquiterpenoid Oxyphyllin A/Belchinoid A
Koichiro Ota, Naoya Kashima, Haruhiko Fukaya, Shinnosuke Okazaki, and Hiroaki Miyaoka
Regular Article
Evaluation of STAT3 Inhibition by Cancer Chemopreventive Trichothecenes Derived from Metabolites of Trichothecium roseum
Mitsuaki Yamashita, Akari Nakanishi, Chiehming Chang, Kosei Tsurushima, Kiyoshige Nakamoto, and Akira Iida
Two Preparation Methods for Peptide Thioester Containing Tyr(SO3H) Residue(s) without the Use of Protecting Group for Sulfate Moiety
Yumi Sekigawa, Shinichi Asada, Yurie Ichikawa, Kazuaki Tsubokawa, Shoh Watanabe, Shinobu Honzawa, and Kouki Kitagawa
Structure-Activity Relationship Study of CYM51010, an Agonist for the µ-δ Opioid Receptor Heterodimer
Ayaka Watanabe, Shuma Yamada, Haruka Yoshida, Miku Inagaki, Nao Atsumi, Aoba Matsushima, Naoki Takahashi, Naoto Ishibashi, Takumi Ogino, Ryoto Someya, Ai Taguchi, Ryo Kagaya, Karin Ashizawa, Hinako Mendori, Yusuke Karasawa, Kaori Ohshima, Akinobu Yokoyama, Miki Nonaka, Kanako Miyano, Fumika Karaki, Shigeto Hirayama, Kennosuke Itoh, Yasuhito Uezono, and Hideaki Fujii
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