NEWS & TOPICS
Chem. Pharm. Bull. Vol. 72 No. 2
2024/04/01
Cover
Advanced Medicinal Chemistry in Academia
pp. 135
Advanced Medicinal Chemistry in Academia
pp. 135
Current Topics - Advanced Medicinal Chemistry in Academia
Foreword
Takayoshi SuzukiCurrent Topics: Review
Targeted Therapy for Prostate Cancer by Prostate-Specific Membrane Antigen-Targeted Small-Molecule Drug Conjugates
Ryo Nakajima
Current Topics: Regular Article
Synthesis of Coumarin-Conjugated Oligonucleotides via Knoevenagel Condensation to Prepare an Oligonucleotide Library
Takashi Osawa and Satoshi Obika
Rational Design of Amphipathic Antimicrobial Peptides with Alternating L-/D-Amino Acids That Form Helical Structures
Motoharu Hirano, Hidetomo Yokoo, Nobumichi Ohoka, Takahito Ito, Takashi Misawa, Makoto Oba, Takao Inoue, and Yosuke Demizu
A Structure-Activity Relationship Study of SNAIL1 Peptides as Inhibitors of Lysine-Specific Demethylase 1
Yuri Takada, Kyohei Adachi, Yuka Fujinaga, Yasunobu Yamashita, Yukihiro Itoh, and Takayoshi Suzuki
Allosteric Hsp70 Modulator YM-1 Induces Degradation of BRD4
Yugo Mishima, Shusuke Tomoshige, Shinichi Sato, and Minoru Ishikawa
In Silico Prediction of N-Nitrosamine Formation Pathways of Pharmaceutical Products
Genichiro Tsuji, Takashi Kurohara, Takuji Shoda, Hidetomo Yokoo, Takahito Ito, Sayaka Masada, Nahoko Uchiyama, Eiichi Yamamoto, and Yosuke Demizu
Identification of a Histone Deacetylase 8 Inhibitor through Drug Screenings Based on Machine Learning
Atika Nurani, Yasunobu Yamashita, Yuuki Taki, Yuri Takada, Yukihiro Itoh, and Takayoshi Suzuki
Note
Total Synthesis of Marine Polyketide Plakortone Q
Shinnosuke Okazaki, Kaho Senda, Ayaka Tokuta, Misa Inagaki, Kazuo Kamaike, Koichiro Ota, and Hiroaki Miyaoka
Sulfonate Derivatives Containing a Kakuol Moiety as Potential Fungicidal Candidates: Design, Synthesis and Antifungal Activity Evaluation
Guoqing Sui, Lili Shu, Ailing Zhang, Dan Li, and Shuhua Cao
Regular Article
Improved Dissolution Properties of Co-amorphous Probucol with Atorvastatin Calcium Trihydrate Prepared by Spray-Drying
Shinji Oyama, Noriko Ogawa, Kaori Kawai, Kanako Iwai, Toshiya Yasunaga, and Hiromitsu Yamamoto
Antiproliferative Activities of Cynaropicrin and Related Compounds against Cancer Stem Cells
Kousuke Araki, Minami Hara, Shohei Hamada, Takahiro Matsumoto, and Seikou Nakamura
Note
Enhanced Physical Stability of L-Ascorbic Acid in an Ionic Liquid
Takeshi Oshizaka, Issei Takeuchi, Katsuya Mukae, Kenji Mori, and Kenji Sugibayashi
Regular Article
Nucleophilic Deprotection of p-Methoxybenzyl Ethers Using Heterogeneous Oxovanadium Catalyst
Rei Ikeda, Tomoya Nishio, Kyohei Kanomata, and Shuji Akai
Note
Effect of Ag and Ni-Doped Cerium Oxide Nanoparticles on the Formation of ROS and Evaluation as an Alternative Physical Sunscreen Material
Agnes Giovanni Marsius, Satria Hidayat, Damar Rastri Adhika, Akhmad Zein Eko Mustofa, Veinardi Suendo, and Heni Rachmawati
Regular Article
Development of a Water Soluble Self-assembling Analogue of Vizantin
Mayo Nakano, Kyohei Sakamoto, Naoto Yamasaki, Yui Asano, Masataka Oda, Hironobu Takahashi, Takashige Kawakami, Masahisa Inoue, and Hirofumi Yamamoto
8-Iodoisoquinolinone, a Conformationally Rigid Highly Reactive 2-Iodobenzamide Catalyst for the Oxidation of Alcohols by Hypervalent Iodine
Takayuki Yakura, Tomoya Fujiwara, Kanna Asakubo, Hema Naga Lakshmi Perumalla, Mitsuha Uzu, Takashi Okitsu, Kengo Kasama, and Hisanori Nambu
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