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NEWS & TOPICS

Chem. Pharm. Bull. Vol. 72 No. 1

2024/03/04

Review

Dual Engineering of Olivetolic Acid Cyclase and Tetraketide Synthase for the Formation of Longer Alkyl-Chain Olivetolic Acid Analogs and Their Antibacterial Activities

Hiroyuki Morita

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Regular Articles

Elucidation of Degradation Behavior of Nitrazepam, a Benzodiazepine Drug, under Basic Conditions: Study on Degradability of Drugs in Stomach (IV)

Koichi Saito, Mai Yokota, Rie Ito, Miho Sakamoto, and Kimio Higashiyama



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Note

Development of an Artificial Nucleic Acid Skeleton Allowing for Unnatural-Type Triplex DNA Formation with Duplex DNA Having a TA Inversion Site

Akihiro Ito, Lei Wang, Ryotaro Notomi, Shigeki Sasaki, and Yosuke Taniguchi

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Regular Article

Preparation and in Vitro Characterization of Fatty-Acid Modified Pirarubicin Nanosuspensions Stabilized by Albumin

Takashi Hasegawa, Kenji Tsukigawa, Kindness Commey, Mina Sakuragi, Shuhei Imoto, Kazuaki Taguchi, Koji Nishi, Masaki Otagiri, and Keishi Yamasaki

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Analysis of Factors Related to Variation in Dissolution Profiles Estimated from Continuously Conducted Dissolution Tests of Generic Products

Tokio Morita, Hiroyuki Yoshida, Yasuhiro Abe, Koji Tomita, Akihiko Nakamura, Chikako Hada, Chiyori Nakai, Keishi Kina, Makoto Takahashi, Nozomi Uemura, Tetsuya Yoneda, Maki Yasui, Yoriko Shintani, Naomi Tomita, Aoi Inagaki, Ken-ichi Izutsu, and Yoji Sato

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Note

Quantitative 31P-NMR for the Purity Determination of the Organophosphorus Compound Brigatinib and Its Method Validation

Nahoko Uchiyama, Junko Hosoe, Takanori Komatsu, Naoki Sugimoto, Kyoko Ishizuki, Tatsuo Koide, Mika Murabayashi, Taeko Shinozaki, Kengo Kobayashi, Yoshinori Fujimine, Katsuya Ofuji, Hitoshi Shimizu, Takashi Hasebe, Yumi Asai, Eri Ena, Kohei Kiyota, Kazuhiro Fujita, Yoshinobu Makino, Toru Miura, Yasuhiro Muto, Katsuo Asakura, Takako Suematsu, Hitomi Muto, Ai Kohama, Takashi Goto, Masu Yasuda, Tomohiko Ueda, and Yukihiro Goda

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Regular Article

Development of Small-Molecule Anti-HIV-1 Agents Targeting HIV-1 Capsid Proteins

Takuya Kobayakawa, Masaru Yokoyama, Kohei Tsuji, Sayaka Boku, Masaki Kurakami, Masayuki Fujino, Takahiro Ishii, Yutaro Miura, Soshi Nishimura, Kouki Shinohara, Kenichi Yamamoto, Peter Bolah, Osamu Kotani, Tsutomu Murakami, Hironori Sato, and Hirokazu Tamamura

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Development of Fast Disintegrating Tablets Containing Loxoprofen Sodium by HYDROFLASH Manufacturing Method

Aya Kuwata, Tetsuo Ono, Yuri Tsuchiya, and Etsuo Yonemochi

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Synthesis of 2,8-Dioxabicyclo[3.3.1]nonane Derivatives and Their Neuroprotective Activities

Hitoshi Kamauchi, Akifumi Takanashi, Mitsuaki Suzuki, Kouki Izumi, Koichi Takao, and Yoshiaki Sugita


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Syntheses and Cytotoxicities of Quinazolinone-Based Conjugates

Hieu Trong Le, Kiep Minh Do, Quy Phu Nguyen, Chau Nguyen Minh Doan, Nhi Ai Nguyen, Tai Thi Phan, Xuyen Thi Cam Tran, Quy Thi Kim Ha, De Quang Tran, Hiroyuki Morita, and Hue Thi Buu Bui

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Bioinspired Total Synthesis of (+)-Kopsiyunnanine B

Sho Imaoka, Yuta Nakashima, Mariko Kitajima, and Hayato Ishikawa

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Efficient and Environmentally Benign Oxidative Cleavage of Pyrrolidine-2-methanols to γ-Lactams Using 2-Iodobenzamide as a Catalyst and Oxone

Hema Naga Lakshmi Perumalla, Tomoya Fujiwara, Maki Okada, Kanna Asakubo, Takashi Okitsu, Kengo Kasama, Hisanori Nambu, and Takayuki Yakura

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Five New Analogs of Streptogramin Antibiotic Viridogrisein Isolated from Streptomyces niveoruber

Aya Yoshimura, Takumi Honda, and Toshiyuki Wakimoto

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Derivation of the Extended Kawakita Equation for Estimating the Yield State of Powder in Die

Tsubasa Sato, Naoto Morita, Etsuo Yonemochi, and Kozo Takayama

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Chromatographic Evaluation and Characterization of Constituents of Sunflower Seed Extract Used as Food Additives

Yoshiaki Amakura, Takashi Uchikura, Morio Yoshimura, Naoko Masumoto, Yuzo Nishizaki, and Naoki

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Note

A Tricyclic Aromatic Polyketide Isolated from the Marine-Derived Fungus Curvularia aeria

Hitoshi Kamauchi, Mayu Tanaka, Mitsuaki Suzuki, Miho Furukawa, Atsushi Ikeda, Chihiro Sasho, Yuka Kiba, Masashi Kitamura, Koichi Takao, and Yoshiaki Sugita

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Regular Article

Development of Ethylcellulose Microparticles for Taste Masking of Fexofenadine

Yuri Ikeuchi-Takahashi, Machi Morii, Kurumi Yamazaki, Aoi Shimana, Ikki Shibazaki, and Yasuko Obata

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Synthesis and Biological Evaluation of 2-Azolylmethylene-3-(2H)-benzofuranone Derivatives as Potent Monoamine Oxidases Inhibitors

Koichi Takao, Yuka Kubota, Kota Kurosaki, Hitoshi Kamauchi, Yoshihiro Uesawa, and Yoshiaki Sugita

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Near-Infrared Fluorescent Silica Nanoparticles Based on Gold-Silver Alloy Nanoclusters for Clinical Diagnosis

Hiroaki Ichimaru and Shigetoshi Kikuchi

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Design, Synthesis, and Biological Evaluation of Water-Soluble Prodrugs of C5-Curcuminoid GO-Y030 Based on Reversible Thia-Michael Reaction

Hiroyuki Yamakoshi, Michihiro Fukuda, Hiro Ikeda, Shogo Fujiki, Aki Kohyama, Shota Nagasawa, Hanae Shinozaki, Hiroyuki Shibata, and Yoshiharu Iwabuchi

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