NEWS & TOPICS
Chem. Pharm. Bull. Vol. 72 No. 1
2024/03/04
Review
Dual Engineering of Olivetolic Acid Cyclase and Tetraketide Synthase for the Formation of Longer Alkyl-Chain Olivetolic Acid Analogs and Their Antibacterial Activities
Hiroyuki Morita
Regular Articles
Elucidation of Degradation Behavior of Nitrazepam, a Benzodiazepine Drug, under Basic Conditions: Study on Degradability of Drugs in Stomach (IV)
Koichi Saito, Mai Yokota, Rie Ito, Miho Sakamoto, and Kimio Higashiyama
Note
Development of an Artificial Nucleic Acid Skeleton Allowing for Unnatural-Type Triplex DNA Formation with Duplex DNA Having a TA Inversion Site
Akihiro Ito, Lei Wang, Ryotaro Notomi, Shigeki Sasaki, and Yosuke Taniguchi
Regular Article
Preparation and in Vitro Characterization of Fatty-Acid Modified Pirarubicin Nanosuspensions Stabilized by Albumin
Takashi Hasegawa, Kenji Tsukigawa, Kindness Commey, Mina Sakuragi, Shuhei Imoto, Kazuaki Taguchi, Koji Nishi, Masaki Otagiri, and Keishi Yamasaki
Analysis of Factors Related to Variation in Dissolution Profiles Estimated from Continuously Conducted Dissolution Tests of Generic Products
Tokio Morita, Hiroyuki Yoshida, Yasuhiro Abe, Koji Tomita, Akihiko Nakamura, Chikako Hada, Chiyori Nakai, Keishi Kina, Makoto Takahashi, Nozomi Uemura, Tetsuya Yoneda, Maki Yasui, Yoriko Shintani, Naomi Tomita, Aoi Inagaki, Ken-ichi Izutsu, and Yoji Sato
Note
Quantitative 31P-NMR for the Purity Determination of the Organophosphorus Compound Brigatinib and Its Method Validation
Nahoko Uchiyama, Junko Hosoe, Takanori Komatsu, Naoki Sugimoto, Kyoko Ishizuki, Tatsuo Koide, Mika Murabayashi, Taeko Shinozaki, Kengo Kobayashi, Yoshinori Fujimine, Katsuya Ofuji, Hitoshi Shimizu, Takashi Hasebe, Yumi Asai, Eri Ena, Kohei Kiyota, Kazuhiro Fujita, Yoshinobu Makino, Toru Miura, Yasuhiro Muto, Katsuo Asakura, Takako Suematsu, Hitomi Muto, Ai Kohama, Takashi Goto, Masu Yasuda, Tomohiko Ueda, and Yukihiro Goda
Regular Article
Development of Small-Molecule Anti-HIV-1 Agents Targeting HIV-1 Capsid Proteins
Takuya Kobayakawa, Masaru Yokoyama, Kohei Tsuji, Sayaka Boku, Masaki Kurakami, Masayuki Fujino, Takahiro Ishii, Yutaro Miura, Soshi Nishimura, Kouki Shinohara, Kenichi Yamamoto, Peter Bolah, Osamu Kotani, Tsutomu Murakami, Hironori Sato, and Hirokazu Tamamura
Development of Fast Disintegrating Tablets Containing Loxoprofen Sodium by HYDROFLASH Manufacturing Method
Aya Kuwata, Tetsuo Ono, Yuri Tsuchiya, and Etsuo Yonemochi
Synthesis of 2,8-Dioxabicyclo[3.3.1]nonane Derivatives and Their Neuroprotective Activities
Hitoshi Kamauchi, Akifumi Takanashi, Mitsuaki Suzuki, Kouki Izumi, Koichi Takao, and Yoshiaki Sugita
Syntheses and Cytotoxicities of Quinazolinone-Based Conjugates
Hieu Trong Le, Kiep Minh Do, Quy Phu Nguyen, Chau Nguyen Minh Doan, Nhi Ai Nguyen, Tai Thi Phan, Xuyen Thi Cam Tran, Quy Thi Kim Ha, De Quang Tran, Hiroyuki Morita, and Hue Thi Buu Bui
Bioinspired Total Synthesis of (+)-Kopsiyunnanine B
Sho Imaoka, Yuta Nakashima, Mariko Kitajima, and Hayato Ishikawa
Efficient and Environmentally Benign Oxidative Cleavage of Pyrrolidine-2-methanols to γ-Lactams Using 2-Iodobenzamide as a Catalyst and Oxone
Hema Naga Lakshmi Perumalla, Tomoya Fujiwara, Maki Okada, Kanna Asakubo, Takashi Okitsu, Kengo Kasama, Hisanori Nambu, and Takayuki Yakura
Five New Analogs of Streptogramin Antibiotic Viridogrisein Isolated from Streptomyces niveoruber
Aya Yoshimura, Takumi Honda, and Toshiyuki Wakimoto
Derivation of the Extended Kawakita Equation for Estimating the Yield State of Powder in Die
Tsubasa Sato, Naoto Morita, Etsuo Yonemochi, and Kozo Takayama
Chromatographic Evaluation and Characterization of Constituents of Sunflower Seed Extract Used as Food Additives
Yoshiaki Amakura, Takashi Uchikura, Morio Yoshimura, Naoko Masumoto, Yuzo Nishizaki, and Naoki
Note
A Tricyclic Aromatic Polyketide Isolated from the Marine-Derived Fungus Curvularia aeria
Hitoshi Kamauchi, Mayu Tanaka, Mitsuaki Suzuki, Miho Furukawa, Atsushi Ikeda, Chihiro Sasho, Yuka Kiba, Masashi Kitamura, Koichi Takao, and Yoshiaki Sugita
Regular Article
Development of Ethylcellulose Microparticles for Taste Masking of Fexofenadine
Yuri Ikeuchi-Takahashi, Machi Morii, Kurumi Yamazaki, Aoi Shimana, Ikki Shibazaki, and Yasuko Obata
Synthesis and Biological Evaluation of 2-Azolylmethylene-3-(2H)-benzofuranone Derivatives as Potent Monoamine Oxidases Inhibitors
Koichi Takao, Yuka Kubota, Kota Kurosaki, Hitoshi Kamauchi, Yoshihiro Uesawa, and Yoshiaki Sugita
Near-Infrared Fluorescent Silica Nanoparticles Based on Gold-Silver Alloy Nanoclusters for Clinical Diagnosis
Hiroaki Ichimaru and Shigetoshi Kikuchi
Design, Synthesis, and Biological Evaluation of Water-Soluble Prodrugs of C5-Curcuminoid GO-Y030 Based on Reversible Thia-Michael Reaction
Hiroyuki Yamakoshi, Michihiro Fukuda, Hiro Ikeda, Shogo Fujiki, Aki Kohyama, Shota Nagasawa, Hanae Shinozaki, Hiroyuki Shibata, and Yoshiharu Iwabuchi
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