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NEWS & TOPICS

Chem. Pharm. Bull. Vol. 71 No. 7

2023/07/03

表紙
Novel Strategies for Enantio- and Site-Selective Molecular Transformations
pp. 466-484

Graphical Abstracts


Review

Novel Strategies for Enantio- and Site-Selective Molecular Transformations

Takeo Kawabata

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Current Topics - Development of Naturally Occurring Compounds for the Treatment of Intractable Diseases

Foreword

Seikou Nakamura

Current Topics: Review

Computer Science Technology in Natural Products Research: A Review of Its Applications and Implications

Keiko Ogawa, Daiki Sakamoto, and Rumiko Hosoki

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Current Topics: Regular Articles

Chemical Structures and Anti-proliferative Effects of Valeriana fauriei Constituents on Cancer Stem Cells

Takahiro Matsumoto, Hayato Yoshikawa, Takahiro Kitagawa, Daisuke Imahori, Tomoe Ohta, Tatsusada Yoshida, and Tetsushi Watanabe

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Antiproliferative Activities of Diterpenes from Leaves of Isodon trichocarpus against Cancer Stem Cells

Seikou Nakamura, Sachiko Sugimoto, Taichi Yoneda, Akari Shinozaki, Moe Yoshiji, Takahiro Matsumoto, Souichi Nakashima, and Hisashi Matsuda

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Angiotensin I-Converting Enzyme-Inhibitory Activity and Phytochemical Profile of Constituents of the Leaves of Rehmannia glutinosa f. hueichingensis

Tomoe Ohta, Momoka Inoha, Chiaki Kawahara, Saori Toshimitsu, Yukihiro Shoyama, and Takuhiro Uto

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Regioselective SmI2-Mediated Radical ipso-Substitution Cyclization for the Construction of Pyrrolophenanthridinone Skeletons: The Synthesis of Amaryllidaceae Alkaloids

Hiroki Iwasaki, Mari Ikemoto, Haruka Shibata, Yuka Shima, Erina Himeno, Naoto Kojima, Masayuki Yamashita, and Hisanori Nambu

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Regular Articles

Optimization of O/W Emulsion Solvent Evaporation Method for Itraconazole Sustained Release Microspheres

Wenping Wang, Honami Kojima, Ming Gao, Xingbin Yin, Takahiro Uchida, and Jian Ni

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A Facile Raman Spectroscopy Method for Online Monitoring of Crystal Plane Orientation of Favipiravir

Shiyi Tang, Rui Feng, Yanlei Kang, Jianbo Cheng, and Jianguang Zhou

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Concise Syntheses of Microsomal Metabolites of a Potent OXE (Oxoeicosanoid) Receptor Antagonist

Shishir Chourey, Rui Wang, Qiuji Ye, Chintam Nagendra Reddy, Shiyu Sun, Norito Takenaka, William S. Powell, and Joshua Rokach

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Structural Characterization of Zinc(II)/Cobalt(II) Complexes of Chiral N-(Anthracen-9-yl)methyl-N,N-bis(2-picolyl)amine and Evaluation of DNA Photocleavage Activity

Yoshimi Ichimaru, Koichi Kato, Rina Nakatani, Risa Isomura, Kirara Sugiura, Yoshihiro Yamaguchi, Wanchun Jin, Hideki Mizutani, Masanori Imai, Masaaki Kurihara, Mikako Fujita, Masami Otsuka, and Hiromasa Kurosaki

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New Candidate Preservative in Ophthalmic Solution Instead of Benzalkonium Chloride: 1,3-Didecyl-2-methyl Imidazolium Chloride

Takuya Iwasaki, Ryosuke Uchiyama, and Kazuto Nosaka

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Design, Synthesis and Structure-Activity Relationship Studies of Protein Kinase CK2 Inhibitors Containing a Purine Scaffold

Keiji Nishiwaki, Shinya Nakamura, Kenji Yoshioka, Eri Nakagawa, Shiori Nakatani, Masato Tsuyuguchi, Takayoshi Kinoshita, and Isao Nakanishi

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Development of a Simple In-Die Method for Determination of Capping Tendency in Rotary Tableting Machines

Yusuke Imayoshi, Shuji Ohsaki, Hideya Nakamura, and Satoru Watano

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Continuous Monitoring of the Hydration Behavior of Hydrophilic Matrix Tablets Using Time-Domain NMR

Takahiro Tsuji, Takashi Ono, Hiromu Taguchi, Kok Hoong Leong, Yoshihiro Hayashi, Shungo Kumada, Kotaro Okada, and Yoshinori Onuki

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Isosteric Replacement of Ester Linkage of Lysophospholipids with Heteroaromatic Rings Retains Potency and Subtype Selectivity

Masaya Ikubo, Akiharu Uwamizu, Luying Chen, Sho Nakamura, Misa Sayama, Hiroki Kawana, Yuko Otani, Kuniyuki Kano, Asuka Inoue, Junken Aoki, and Tomohiko Ohwada

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Notes

Analysis of Acetylated Hyaluronic Acid in Moisturizing Lotion and Milk Lotion by HPLC with Fluorescence Detection

Momo Shimekake, Masahiro Komeno, Manawo Taguchi, Shoo Katsumoto, Yuna Tanda, Kazuki Sato, Takeshi Wada, Toshihiko Toida, and Kyohei Higashi

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Syntheses of Aryl Thioethers via Aromatic Substitution of Aryl Halides at 0 to 25°C

Marina Tsuzaki, Shin Ando, and Tadao Ishizuka

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