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Chem. Pharm. Bull. Vol. 71 No. 2

2023/02/01

　

表紙

Transition Metal Catalysis Research in Pharmaceutical Organic Chemistrypp. 78-110

Graphical Abstracts

Current Topics - Transition Metal Catalysis Research in Pharmaceutical Organic Chemistry

Foreword

Tetsuhiro Nemoto

Current Topics: Communication to the Editor

Noble-Metal-Free C-H Allylation of Tetrahydroisoquinolines Using a Cobalt-Organophotoredox Dual Catalyst System

Shunta Sato, Wataru Sasaki, Tomoyuki Sekino, Tatsuhiko Yoshino, Masahiro Kojima, and Shigeki Matsunaga

Current Topics: Regular Articles

Copper-Catalyzed Aerobic C(sp³)-H Oxidation of β-(Alkoxy)imino Carbonyl Compounds

Masafumi Ueda, Ayano Ichimonji, Miku Nakayama, Sachiko Ito, Norihiko Takeda, and Motohiro Yasui

Palladium-Catalyzed Intramolecular Migratory Cycloisomerization of 3-Phenoxy Acrylic Acid Ester via C-O Bond Cleavage and C-O/C-C Bonds Formation for 2,3-Disubstituted Benzofurans Synthesis

Yuichi Kuboki, Shohei Ohno, Makoto Sako, Kenichi Murai, and Mitsuhiro Arisawa

O- and N-Selective Electrophilic Activation of Allylic Alcohols and Amines in Pd-Catalyzed Direct Alkylation

Lu Lin, Shunsuke Kataoka, Kiichi Hirayama, Ryozo Shibuya, Kenji Watanabe, Hiroyuki Morimoto, and Takashi Ohshima

Theoretical Investigation of Chemoselectivity between C-H Insertion and Amide Insertion in Intramolecular Rhodium-Carbene Reactions

Tsukasa Furuya, Kotaro Ikeda, Shingo Harada, and Tetsuhiro Nemoto

Regular Articles

Promoting Activity of Terpenes on Skin Permeation of Famotidine

Qihui Xu, Yifan Wu, Hiroki Saito, Yuki Ofuchi, Haruna Setoyama, Takayuki Furuishi, Kaori Fukuzawa, Etsuo Yonemochi, and Yasuko Obata

Design, Synthesis, and Biological Evaluation of mTOR-Targeting PROTACs Based on MLN0128 and Pomalidomide

Qi Zhang, Peizheng Yan, Pan Zhao, Dongsheng Zhao, Heran Cao, Jing Lu, and Beibei Mao

Effects of Emodin on Protein Expression Related to Autophagy of Interstitial Cells of Cajal in Diabetic Rats

Yujin Wang, Na Dong, Yuan Zhou, Hongyan Li, Gangxin Qin, Hui Li, Qiaoqiao Zhao, Miao Zhang, and Yanjin Su

Quantification of Risperidone Contained in Precipitates Produced by Tea Catechins Using Nuclear Magnetic Resonance

Takeshi Goromaru, Kai Fujita, Misaki Mizumoto, and Takashi Ishizu

Synthesis and Evaluation of 2-Amine-4-oxyphosaniline Pyrimidine Derivatives as EGFR L858R/T790M/C797S Mutant Inhibitors

Mingguang Zhang, Yang Yang, Yunyun Wang, Jia Wang, Hongyan Wu, and Yongqiang Zhu

Masking the Taste of Fixed-Dose Combination Drugs: Particular NSAIDs Can Efficiently Mask the Bitterness of Famotidine

Rio Uno, Kyoko Ohkawa, Honami Kojima, Tamami Haraguchi, Minoru Ozeki, Ikuo Kawasaki, Miyako Yoshida, Masaaki Habara, Hidekazu Ikezaki, and Takahiro Uchida

Identification of a Functionally Efficient and Thermally Stable Outward Sodium-Pumping Rhodopsin (BeNaR) from a Thermophilic Bacterium

Marie Kurihara, Vera Thiel, Hirona Takahashi, Keiichi Kojima, David M. Ward, Donald A. Bryant, Makoto Sakai, Susumu Yoshizawa, and Yuki Sudo

Quality Evaluation of Humidified Magnesium Oxide Tablet Formulations with Respect to Disintegration Time Prolongation

Yoshihisa Yamamoto, Kosuke Ohgi, Yoshinori Onuki, Toshiro Fukami, and Tatsuo Koide

Palladium-Catalyzed C-H Arylation of [1,1′-Biphenyl]-2-ols with Chloroarenes

Keisuke Kinoshita, Miyuki Yamaguchi, Hirohisa Sasou, Hideyuki Konishi, and Kei Manabe

Note

Briastecholide M, a New Polyoxygenated Briarane from Briareum stechei

Thanh Hao Huynh, Zhi-Hong Wen, Jui-Hsin Su, Zhi-Kang Yao, Li-Guo Zheng, Yu-Chi Tsai, Junichi Tanaka, Chia-Ching Liaw, and Ping-Jyun Sung

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