NEWS & TOPICS
Chem. Pharm. Bull. Vol. 71 No. 2
2023/02/01
Current Topics - Transition Metal Catalysis Research in Pharmaceutical Organic Chemistry
Foreword
Tetsuhiro Nemoto
Current Topics: Communication to the Editor
Noble-Metal-Free C-H Allylation of Tetrahydroisoquinolines Using a Cobalt-Organophotoredox Dual Catalyst System
Shunta Sato, Wataru Sasaki, Tomoyuki Sekino, Tatsuhiko Yoshino, Masahiro Kojima, and Shigeki Matsunaga
Current Topics: Regular Articles
Copper-Catalyzed Aerobic C(sp3)-H Oxidation of β-(Alkoxy)imino Carbonyl Compounds
Masafumi Ueda, Ayano Ichimonji, Miku Nakayama, Sachiko Ito, Norihiko Takeda, and Motohiro Yasui
Palladium-Catalyzed Intramolecular Migratory Cycloisomerization of 3-Phenoxy Acrylic Acid Ester via C-O Bond Cleavage and C-O/C-C Bonds Formation for 2,3-Disubstituted Benzofurans Synthesis
Yuichi Kuboki, Shohei Ohno, Makoto Sako, Kenichi Murai, and Mitsuhiro Arisawa
O- and N-Selective Electrophilic Activation of Allylic Alcohols and Amines in Pd-Catalyzed Direct Alkylation
Lu Lin, Shunsuke Kataoka, Kiichi Hirayama, Ryozo Shibuya, Kenji Watanabe, Hiroyuki Morimoto, and Takashi Ohshima
Theoretical Investigation of Chemoselectivity between C-H Insertion and Amide Insertion in Intramolecular Rhodium-Carbene Reactions
Tsukasa Furuya, Kotaro Ikeda, Shingo Harada, and Tetsuhiro Nemoto
Regular Articles
Promoting Activity of Terpenes on Skin Permeation of Famotidine
Qihui Xu, Yifan Wu, Hiroki Saito, Yuki Ofuchi, Haruna Setoyama, Takayuki Furuishi, Kaori Fukuzawa, Etsuo Yonemochi, and Yasuko Obata
Design, Synthesis, and Biological Evaluation of mTOR-Targeting PROTACs Based on MLN0128 and Pomalidomide
Qi Zhang, Peizheng Yan, Pan Zhao, Dongsheng Zhao, Heran Cao, Jing Lu, and Beibei Mao
Effects of Emodin on Protein Expression Related to Autophagy of Interstitial Cells of Cajal in Diabetic Rats
Yujin Wang, Na Dong, Yuan Zhou, Hongyan Li, Gangxin Qin, Hui Li, Qiaoqiao Zhao, Miao Zhang, and Yanjin Su
Quantification of Risperidone Contained in Precipitates Produced by Tea Catechins Using Nuclear Magnetic Resonance
Takeshi Goromaru, Kai Fujita, Misaki Mizumoto, and Takashi Ishizu
Synthesis and Evaluation of 2-Amine-4-oxyphosaniline Pyrimidine Derivatives as EGFR L858R/T790M/C797S Mutant Inhibitors
Mingguang Zhang, Yang Yang, Yunyun Wang, Jia Wang, Hongyan Wu, and Yongqiang Zhu
Masking the Taste of Fixed-Dose Combination Drugs: Particular NSAIDs Can Efficiently Mask the Bitterness of Famotidine
Rio Uno, Kyoko Ohkawa, Honami Kojima, Tamami Haraguchi, Minoru Ozeki, Ikuo Kawasaki, Miyako Yoshida, Masaaki Habara, Hidekazu Ikezaki, and Takahiro Uchida
Identification of a Functionally Efficient and Thermally Stable Outward Sodium-Pumping Rhodopsin (BeNaR) from a Thermophilic Bacterium
Marie Kurihara, Vera Thiel, Hirona Takahashi, Keiichi Kojima, David M. Ward, Donald A. Bryant, Makoto Sakai, Susumu Yoshizawa, and Yuki Sudo
Quality Evaluation of Humidified Magnesium Oxide Tablet Formulations with Respect to Disintegration Time Prolongation
Yoshihisa Yamamoto, Kosuke Ohgi, Yoshinori Onuki, Toshiro Fukami, and Tatsuo Koide
Palladium-Catalyzed C-H Arylation of [1,1′-Biphenyl]-2-ols with Chloroarenes
Keisuke Kinoshita, Miyuki Yamaguchi, Hirohisa Sasou, Hideyuki Konishi, and Kei Manabe
Note
Briastecholide M, a New Polyoxygenated Briarane from Briareum stechei
Thanh Hao Huynh, Zhi-Hong Wen, Jui-Hsin Su, Zhi-Kang Yao, Li-Guo Zheng, Yu-Chi Tsai, Junichi Tanaka, Chia-Ching Liaw, and Ping-Jyun Sung
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