ABSTRACT ABSTRACT 29-413-pm03S Structure-activity relationship (SAR) study of hydrophobic moiety of nonsecosteroidal VDR ligands using diphenylsilane scaffold ○Hansaka Nirupama Thilakarathne Narasinghe Mudiyanselage1,2, Takashi Misawa3, Yosuke Demizu3, Yuya Hanazono2, Nobutoshi Ito2, Hiroyuki Kagechika1, Shinya Fujii1 1. Institute of Biomaterials and Bioengineering, Tokyo medical and Dental Univ., 2. Medical Research Institute, Tokyo Medical and Dental Univ., 3. National Institute of Health Sciences 30-413-pm05S Evaluation of Target Protein Degradation Activity and Physicochemical Properties of Trivalent PROTACs Based on Brd4 Degrader MZ1 ○Yifan Huang1, Marina Sampei2, Hiromasa Yokoe2,3, Fumiaki Ohtake2,4, Naoki Kanoh2,3 1. Graduate Sch. Pharmaceut. Sci., Hoshi Univ., 2. Sch. Pharm. and Pharmaceut. Sci., Hoshi Univ., 3. Institute of Medicinal Chemistry, Hoshi Univ., 4. Institute for Advanced Life Sciences, Hoshi Univ. ABSTRACT 30-413-pm10 Targeting transcription factors with PROTACS: the FOXM1 protein ○Carlos A Velázquez1, Gordon Chan2, Adam Karpf3, Antonio Vega-Medina1, Erika Loredo-Calderon1 1. Fac. Pharm. & Pharm. Sci., U. of A., 2. Fac. Med. Dent., U. of A., 3. Univ. Nebraska, Med. Centre. 31-413-am03S Discovery of hydrophobic tag-based degraders targeting lysine-specific demethylase 1 ○SHENGWANG YU1, Yasunobu Yamashita1, Yuri Takada1, Yukihiro Itoh1, Takayoshi Suzuki1 1. SANKEN, Osaka Univ. 31-413-am04S Enhancing T-cell activation: Synthesis of meta-carboranes regulating CD28 binding to SH2 domains of Grb2 and PI3K ○YUJIE SHAO1, Yasunobu Asawa1, Shuhei Ogawa2, Saki Ochi3, Atsushi Yoshimori4, Masayuki Oda3, Hiroyuki Nakamura1,5 1. Sch. Life Sci. & tech., Tokyo Institute of Technology., 2. Research Institute for Biomedical Sciences, Tokyo Univ. Science., 3. Graduate Sch. Life and Environmental Sciences, Kyoto Prefectural Univ., 4. Institute for Theoretical Medicine, Inc., 5. Institute of Innovative Research, Tokyo Institute of Technology 31-413-am05 Direct Catalytic Enantioselective Conjugate Addition of α-Substituted Benzyl ○Yingchao Wang1,2, Kouharu Otsuki1, Bingyang Zhang2, Tie Yao2, Takashi Kikuchi1, Feng Qiu2, Wei Li1 1. Fac. Pharm. Sci., Toho Univ., 2. Tianjin Univ. Traditional Chinese Medicine ABSTRACT ABSTRACT ABSTRACT
元のページ ../index.html#23